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Inhibitor Libraries
  PIM1 Inhibitor II
Cat. No. 526520  
All Categories » Calbiochem » Inhibitors » Kinase and Phosphatase » PIM Kinase

3-Cyano-4-phenyl-6-(3-bromo-6-hydroxy)phenyl-2(1H)-pyridone
2-Hydroxy-3-cyano-4-phenyl-6-(3-bromo-6-hydroxyphenyl)pyridine

Yellow solid. PROTECT FROM LIGHT. PACKAGED UNDER INERT GAS. A pyridone compound that acts as an ATP-competitive inhibitor of PIM1 kinase (IC50 = 50 nM) with excellent selectivity over PIM2 and MEK1/2 (IC50 > 20 µM). Purity: ≥90% by HPLC.

Ref.: Cheney, I. W., et al. 2007. Bioorg. Med. Chem. Lett. 17, 1679.

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5 mgY$96.00

SolubilityMolecular FormulaMol. Wt.
DMSO C18H11BrN2O2 367.2 


Material Safety Data Sheets:
526520: PIM1 Inhibitor II - English

Related Categories:
All Categories » Calbiochem » Inhibitors » Kinase and Phosphatase » PIM Kinase